GHRP-6 5MG

$19.99

GHRP 6 for sale is available in lyophilized powder form, in 5mg vials.

SKU: ghrp6 Category: Tags: ,

Description

About GHRP-6: GHRP-6 is a synthetic growth hormone (GH) secretagogue and an agonist of the GH secretagogue receptor (GHS-R), which is also known as the ghrelin receptor.1,2,3,4 It inhibits binding of the GHS-R agonist MK-0677 (ibutamoren) to COS-7 cell membranes expressing human GHS-R type Ia (Ki = 1.9 nM) and binding of ghrelin to COS-7 cells expressing human GHS-R (Kd = 260 nM).2,3

GHRP-6 stimulates intracellular calcium mobilization in BHK cells expressing the human receptor (EC50 = 4.5 nM) and inositol phosphate production in COS-7 cells expressing the human receptor (EC50 = 0.83 nM).3 It also acts as a negative allosteric modulator of ghrelin signaling. GHRP-6 (0.03 μg/ml) induces release of GH, but not thyroid-stimulating hormone (TSH), luteinizing hormone (LH), or follicle-stimulating hormone (FSH), in isolated rat pituitary gland.1

It increases levels of GH, but not TSH, LH, FSH, or prolactin, in rat blood when administered subcutaneously at a dose of 50 μg. GHRP-6 increases food intake in rats when administered intracerebroventricularly at 0.3, 1, and 3 nmol.4

BUY GHRP-6 Today from GenX Peptides.

We offer the highest grade and purity of GHRP 6 for sale at a competitive price in the USA. For best results buy GHRP-6 of the highest quality from GenX Peptides.

For more information on GHRP-6 5mg peptide please visit Pubmed.

References & Product Citations

Product Description References

1. Bowers, C.Y., Momany, F.A., Reynolds, G.A., et al. On the in vitro and in vivo activity of a new synthetic hexapeptide that acts on the pituitary to specifically release growth hormone. Endocrinology 114(5), 1537-1545 (1984).

2. Howard, A.D., Feighner, S.D., Cully, D.F., et al. A receptor in pituitary and hypothalamus that functions in growth hormone release. Science 273(5277), 974-977 (1996).

3. Holst, B., Brandt, E., Bach, A., et al. Nonpeptide and peptide growth hormone secretagogues act both as ghrelin receptor agonist and as positive or negative allosteric modulators of ghrelin signaling. Mol. Endocrinol. 19(9), 2400-2411 (2005).

4. Wren, A.M., Small, C.J., Ward, H.L., et al. The novel hypothalamic peptide ghrelin stimulates food intake and growth hormone secretion. Endocrinology 141(11), 4325-4328 (2000).

Unit Size5 mg/vial
Unit Quantity1 Vial
Molecular FormulaC46H56N12O6
Molecular Weight873.04
SequenceH-His-D-Trp-Ala-Trp-D-Phe-Lys-NH2
AppearanceWhite Powder
Peptide Purity>99%
Solubility>Soluble in water or 1% acetic acid
Identity (ESI-MS)873.01±1.0
SourceChemical Synthesis
StorageLyophilized GHRP-6 is stable at room temperature for 90 days, however it should be stored in a freezer below -8C for any extended period of time.
Safety InformationFor Research Only. Not Intended for Diagnostic or Therapeutic Use.

Additional information

Weight1 oz
Dimensions1 × 1 × 1 in

Content missing

GHRP 6 Peptide Vial
GHRP-6 5MG
$19.99
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