GW1516 Cardarine 30mL 10mg/mL

Name: GW501516 Cardarine 30mL 10mg/mL
Brand: Liquids
SKU: gw501516
Price: 44.99 USD
Availability: InStock

$44.99

GW 501516 for sale is available in 30mL liquid form.

In stock

Full description

SKU: gw501516 Category: Liquids Tag: SARMs

Description
Additional information

Description

About GW-501516: Peroxisome proliferator-activated receptor δ (PPARδ) stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity.¹ GW 501516 is the first highly selective synthetic PPARδ agonist available. GW 501516 binds to human PPARδ with an IC₅₀ value of 1 nM, and is at least 100-fold selective for PPARδ compared to PPARα and PPARγ.² In obese primates, GW 501516 increases high density lipoprotein cholesterol and apolipoprotein A-1 specific reverse cholesterol transport.³ GW 501516 is therefore a model compound for a new type of obesity therapeutic, as well as a selective pharmacological tool for understanding lipid metabolism.

Buy GW-501516 Today from GenX Peptides.

We offer the highest grade and purity of GW501516 for sale at a competitive price in the USA. For best results buy GW 501516 of the highest quality from GenX Peptides.

For more information on Endurobol PPARδ receptor agonist please visit Pubmed.

References & Product Citations

Product Description References

1. Wang, Y.X., Lee, C.H., Tiep, S., et al. Peroxisome-proliferator-activated receptor δ activates fat metabolism to prevent obesity. Cell 113, 159-170 (2003).

2. Sznaidman, M.L., Haffner, C.D., Maloney, P.R., et al. Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)-synthesis and biological activity. Bioorg. Med. Chem. Lett. 13(9), 1517-1521 (2003).

3. Oliver, W.R., Shenk, J.L., Snaith, M.R., et al. A selective peroxisome proliferator-activated receptor δ agonist promotes reverse cholesterol transport. Proceedings of the National Academy of Sciences of the United States of America 98(9), 5306-5311 (2001).

Product Citations

Wang, X., Wang, G., Shi, Y., et al. PPAR-delta promotes survival of breast cancer cells in harsh metabolic conditions. Oncogenesis 5, e232 (2016).

Concentration: 10mg per mL, 300mg/30mL total

Description

Read the Cardarine Specification Before Buying:

Application	PPARδ receptor agonist
CAS	317318-70-0
Molar Mass	453.498 g/mol
Chemical Formula	C₂₁H₁₈F₃NO₃S₂
Chemical Name	{4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]-2-methylphenoxy}acetic acid
Synonyms	GW501516, Cardarine, Endurobol, GSK-516
Storage	Room temperature
Solubility	PEG, Ethanol
Organoleptic Profile	Clear Liquid
Physical Form	Solution in PEG-400, Ethanol (0.5%)
Safety Information	For Research Only. Not for Diagnostic or Therapeutic use