GW501516 Cardarine 30mL 10mg/mL

$44.99

GW 501516 for sale is available in 30mL liquid form.

SKU: gw501516 Category: Tag:

Description

About GW-501516: Peroxisome proliferator-activated receptor δ (PPARδ) stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity.1 GW 501516 is the first highly selective synthetic PPARδ agonist available. GW 501516 binds to human PPARδ with an IC50 value of 1 nM, and is at least 100-fold selective for PPARδ compared to PPARα and PPARγ.2 In obese primates, GW 501516 increases high density lipoprotein cholesterol and apolipoprotein A-1 specific reverse cholesterol transport.3 GW 501516 is therefore a model compound for a new type of obesity therapeutic, as well as a selective pharmacological tool for understanding lipid metabolism.

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We offer the highest grade and purity of GW501516 for sale at a competitive price in the USA. For best results buy GW 501516 of the highest quality from GenX Peptides.

For more information on Endurobol PPARδ receptor agonist please visit Pubmed.

References & Product Citations

Product Description References

1. Wang, Y.X., Lee, C.H., Tiep, S., et al. Peroxisome-proliferator-activated receptor δ activates fat metabolism to prevent obesity. Cell 113, 159-170 (2003).

2. Sznaidman, M.L., Haffner, C.D., Maloney, P.R., et al. Novel selective small molecule agonists for peroxisome proliferator-activated receptor δ (PPARδ)-synthesis and biological activity. Bioorg. Med. Chem. Lett. 13(9), 1517-1521 (2003).

3. Oliver, W.R., Shenk, J.L., Snaith, M.R., et al. A selective peroxisome proliferator-activated receptor δ agonist promotes reverse cholesterol transport. Proceedings of the National Academy of Sciences of the United States of America 98(9), 5306-5311 (2001).

Product Citations

Wang, X., Wang, G., Shi, Y., et al. PPAR-delta promotes survival of breast cancer cells in harsh metabolic conditions. Oncogenesis 5, e232 (2016).

Concentration: 10mg per mL, 300mg/30mL total

  • Description

Read the Cardarine Specification Before Buying:

ApplicationPPARδ receptor agonist
CAS317318-70-0
Molar Mass453.498 g/mol
 Chemical FormulaC21H18F3NO3S2
Chemical Name{4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]-2-methylphenoxy}acetic acid
SynonymsGW501516, Cardarine, Endurobol, GSK-516
StorageRoom temperature
SolubilityPEG, Ethanol
Organoleptic ProfileClear Liquid
Physical FormSolution in PEG-400, Ethanol (0.5%)
Safety InformationFor Research Only. Not for Diagnostic or Therapeutic use

Additional information

Weight1 oz
Dimensions1 × 1 × 2 in
buy cardarine (GW-501516)
GW501516 Cardarine 30mL 10mg/mL
$44.99
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